Loading...
Derniers dépôts
-
Nathan Picois, Lizeth Bodero, Pierre T Milbeo, Thierry Brigaud, Grégory Chaume. Bimodal use of chiral α‐Trifluoromethylalanine in Aib Foldamers: study of the position impact towards the helical screw‐sense preference. Chemistry - A European Journal, In press, ⟨10.1002/chem.202400540⟩. ⟨hal-04516499⟩
-
Julia Kaffy, Dimitri Brinet, Jean-Louis Soulier, Isabelle Correia, Nicolo Tonali, et al.. Designed Glycopeptidomimetics Disrupt Protein–Protein Interactions Mediating Amyloid β-Peptide Aggregation and Restore Neuroblastoma Cell Viability. Journal of Medicinal Chemistry, 2016, 59 (5), pp.2025-2040. ⟨10.1021/acs.jmedchem.5b01629⟩. ⟨hal-02467871⟩
-
Doumet Georges Helou, A. Mauras, Francois Fasquelle, J. S. Lanza, P. M. Loiseau, et al.. Intranasal vaccine from whole Leishmania donovani antigens provides protection and induces specific immune response against visceral leishmaniasis.. PLoS Neglected Tropical Diseases, 2021, PLoS Neglected Tropical Diseases, 15, pp.e0009627. ⟨10.1371/journal.pntd.0009627⟩. ⟨hal-04482585⟩
Mots-clés
Antiviral
Biological activity
Amphidinolide
Article
Circular dichroism
Glycosides
Enynes
Autoimmune diseases
Benzofuran
Halogenation
Apoptosis
IsoCA-4
Hair
Heterocycles
Peptidomimétiques
Amyloïde
Alkynes
Combretastatin A-4
ACL
Peptidomimetics
Buchwald-Hartwig-Migita coupling
Cancer
High-resolution mass spectrometry
Capillary electrophoresis
Fluorescence
Alteration
Synthetic methods
Aldehydes
Cytotoxicity
NMR
Dereplication
Tubulin
DMSO
Benzils
Thiosugars
Sodium iodide
Mass spectrometry
Hydrostannation
Fluorine
Fluor
Biosynthesis
Molecular networking
Conformational analysis
Environmental neurotoxin
Leishmania
Chalcones
Chitosan
Binding
Amyloid
Annulations
Biotransformation
Autoanticorps
Catalysis
Alkynylation
Glycosylation
Crystallography
Annonacin
Asymmetric synthesis
Human
Peptides
Force-field
Archéométrie des matières colorantes
Palladium
Ribavirin
5-HT 4 receptor
Antileishmanial
Chemical diversity
Antimitotic
Leishmaniasis
Alkyne
Fluorinated peptides
Aggregation
C-nucleoside
Biosynthèse
Cyclization
Alpha-synuclein
CXCR4
Michael addition
Benthic cyanobacteria
Antimicrobial activity
Copper
Autoantibodies
Annonaceae
Antimalarial
Foldamers
Pigments
Natural products
Carbohydrates
Biomimetic synthesis
Controlled study
Constrained amino acids
Coupling
Chemistry
Binding site
Molecular dynamics
Conformational ensemble
Molecular modeling
Acetogenin
Alkaloids
Ilimaquinone